Anxiolytic Peptide

Selank

Tuftsin Analog (TKPRPGP)

Selank — Research Overview

Selank is a synthetic analog of tuftsin, a naturally occurring immunostimulant tetrapeptide. It has been extensively studied in Russia as an anxiolytic agent and is approved there for anxiety and asthenia treatment.

Sequence
Thr-Lys-Pro-Arg-Pro-Gly-Pro
Molecular Weight
751.87 g/mol
Half-life (Preclinical)
~2 minutes (plasma); extended CNS activity
Mechanism
GABAergic modulation; enkephalin degradation inhibition; BDNF expression
Storage
-20°C
Solubility
Water

Research Summary

Published Russian research includes both animal studies and human clinical trials for generalized anxiety. Selank appears to slow enzymatic degradation of endogenous enkephalins and upregulates BDNF expression.

Research Strengths
  • Anxiolytic activity in animal models
  • Immunomodulatory profile
  • Human data exists (Russian trials)
  • Well-characterized mechanism
Limitations & Considerations
  • Extremely short plasma half-life
  • Most research is Russian-language
  • Regulatory status varies by country
This information is for research reference only. Selank is a Research Use Only (RUO) compound not approved for human or veterinary use. This does not constitute medical advice.